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-Structure paper
Title | Highly Selective Phosphatidylinositol 4-Kinase III beta Inhibitors and Structural Insight into Their Mode of Action. |
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Journal, issue, pages | J. Med. Chem., Vol. 58, Page 3767-3793, Year 2015 |
Publish date | Aug 29, 2014 (structure data deposition date) |
Authors | Mejdrova, I. / Chalupska, D. / Kogler, M. / Sala, M. / Plackova, P. / Baumlova, A. / Hrebabecky, H. / Prochazkova, E. / Dejmek, M. / Guillon, R. ...Mejdrova, I. / Chalupska, D. / Kogler, M. / Sala, M. / Plackova, P. / Baumlova, A. / Hrebabecky, H. / Prochazkova, E. / Dejmek, M. / Guillon, R. / Strunin, D. / Weber, J. / Lee, G. / Birkus, G. / Mertlikova-Kaiserova, H. / Boura, E. / Nencka, R. |
External links | J. Med. Chem. / PubMed:25897704 |
Methods | X-ray diffraction |
Resolution | 3.318 - 3.407 Å |
Structure data | PDB-4wae: PDB-4wag: |
Chemicals | ChemComp-ATP: ChemComp-3K7: |
Source |
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Keywords | TRANSFERASE / inhibitor |