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-Structure paper
Title | Engineering of an isolated p110 alpha subunit of PI3K alpha permits crystallization and provides a platform for structure-based drug design. |
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Journal, issue, pages | Protein Sci., Vol. 23, Page 1332-1340, Year 2014 |
Publish date | Jun 24, 2014 (structure data deposition date) |
![]() | Chen, P. / Deng, Y.L. / Bergqvist, S. / Falk, M.D. / Liu, W. / Timofeevski, S. / Brooun, A. |
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Methods | X-ray diffraction |
Resolution | 2.64 - 2.85 Å |
Structure data | ![]() PDB-4tuu: ![]() PDB-4tv3: |
Chemicals | ![]() ChemComp-HOH: ![]() ChemComp-ML9: |
Source |
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![]() | TRANSFERASE / Lipid kinase activity / ATPase activity / Surface Plasmon Resonance (SPR) / isothermal titration calorimetry (ITC). / TRANSFERASE/TRANSFERASE Inhibitor / TRANSFERASE-TRANSFERASE Inhibitor complex |