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-Structure paper
Title | Discovery and profiling of a selective and efficacious syk inhibitor. |
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Journal, issue, pages | J. Med. Chem., Vol. 58, Page 1950-1963, Year 2015 |
Publish date | Dec 9, 2014 (structure data deposition date) |
![]() | Thoma, G. / Smith, A.B. / van Eis, M.J. / Vangrevelinghe, E. / Blanz, J. / Aichholz, R. / Littlewood-Evans, A. / Lee, C.C. / Liu, H. / Zerwes, H.G. |
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Methods | X-ray diffraction |
Resolution | 1.59 - 1.8 Å |
Structure data | ![]() PDB-4rx7: ![]() PDB-4rx8: ![]() PDB-4rx9: |
Chemicals | ![]() ChemComp-FMT: ![]() ChemComp-GOL: ![]() ChemComp-3YV: ![]() ChemComp-HOH: ![]() ChemComp-3YX: ![]() ChemComp-3YT: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / TRANSFERASE-TRANSFERASE INHIBITOR complex |