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-Structure paper
Title | Development of Organometallic S6K1 Inhibitors. |
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Journal, issue, pages | J. Med. Chem., Vol. 58, Page 305-314, Year 2015 |
Publish date | Oct 17, 2014 (structure data deposition date) |
Authors | Qin, J. / Rajaratnam, R. / Feng, L. / Salami, J. / Barber-Rotenberg, J.S. / Domsic, J. / Reyes-Uribe, P. / Liu, H. / Dang, W. / Berger, S.L. ...Qin, J. / Rajaratnam, R. / Feng, L. / Salami, J. / Barber-Rotenberg, J.S. / Domsic, J. / Reyes-Uribe, P. / Liu, H. / Dang, W. / Berger, S.L. / Villanueva, J. / Meggers, E. / Marmorstein, R. |
External links | J. Med. Chem. / PubMed:25356520 |
Methods | X-ray diffraction |
Resolution | 2.527 - 2.79 Å |
Structure data | PDB-4rlo: PDB-4rlp: |
Chemicals | ChemComp-3T3: ChemComp-GOL: ChemComp-CL: ChemComp-SO4: ChemComp-STU: ChemComp-DMS: ChemComp-HOH: ChemComp-72B: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / kinase / TRANSFERASE-TRANSFERASE INHIBITOR complex |