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-Structure paper
Title | Kinase domain inhibition of leucine rich repeat kinase 2 (LRRK2) using a [1,2,4]triazolo[4,3-b]pyridazine scaffold. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 24, Page 4132-4140, Year 2014 |
Publish date | Mar 25, 2014 (structure data deposition date) |
Authors | Galatsis, P. / Henderson, J.L. / Kormos, B.L. / Han, S. / Kurumbail, R.G. / Wager, T.T. / Verhoest, P.R. / Noell, G.S. / Chen, Y. / Needle, E. ...Galatsis, P. / Henderson, J.L. / Kormos, B.L. / Han, S. / Kurumbail, R.G. / Wager, T.T. / Verhoest, P.R. / Noell, G.S. / Chen, Y. / Needle, E. / Berger, Z. / Steyn, S.J. / Houle, C. / Hirst, W.D. |
External links | Bioorg. Med. Chem. Lett. / PubMed:25113930 |
Methods | X-ray diffraction |
Resolution | 2.16 Å |
Structure data | PDB-4py1: |
Chemicals | ChemComp-2YK: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE / kinase |