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| Title | On the metabolically active form of metaglidasen: improved synthesis and investigation of its peculiar activity on peroxisome proliferator-activated receptors and skeletal muscles. |
|---|---|
| Journal, issue, pages | Chemmedchem, Vol. 10, Page 555-565, Year 2015 |
| Publish date | Mar 18, 2014 (structure data deposition date) |
Authors | Laghezza, A. / Montanari, R. / Lavecchia, A. / Piemontese, L. / Pochetti, G. / Iacobazzi, V. / Infantino, V. / Capelli, D. / De Bellis, M. / Liantonio, A. ...Laghezza, A. / Montanari, R. / Lavecchia, A. / Piemontese, L. / Pochetti, G. / Iacobazzi, V. / Infantino, V. / Capelli, D. / De Bellis, M. / Liantonio, A. / Pierno, S. / Tortorella, P. / Conte Camerino, D. / Loiodice, F. |
External links | Chemmedchem / PubMed:25641779 |
| Methods | X-ray diffraction |
| Resolution | 2.6 Å |
| Structure data | ![]() PDB-4pvu: ![]() PDB-4pwl: |
| Chemicals | ![]() ChemComp-MGZ: ![]() ChemComp-HOH: ![]() ChemComp-MSZ: |
| Source |
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Keywords | TRANSCRIPTION / ALPHA-HELICES / SMALL FOUR-STRANDED BETA-SHEET / ACTIVATOR / TDNA-BINDING / NUCLEUS / OBESITY / RECEPTOR / TRANSCRIPTION REGULATION / DNA-BINDING / TRANSCRIPTION REGULATION X-RAY DIFFRACTION / Transcription Factor / RXR-alpha |
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homo sapiens (human)
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