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-Structure paper
Title | Structural Basis for Isoform Selectivity in a Class of Benzothiazole Inhibitors of Phosphoinositide 3-Kinase gamma. |
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Journal, issue, pages | J. Med. Chem., Vol. 58, Page 517-521, Year 2015 |
Publish date | Mar 6, 2014 (structure data deposition date) |
![]() | Collier, P.N. / Martinez-Botella, G. / Cornebise, M. / Cottrell, K.M. / Doran, J.D. / Griffith, J.P. / Mahajan, S. / Maltais, F. / Moody, C.S. / Huck, E.P. ...Collier, P.N. / Martinez-Botella, G. / Cornebise, M. / Cottrell, K.M. / Doran, J.D. / Griffith, J.P. / Mahajan, S. / Maltais, F. / Moody, C.S. / Huck, E.P. / Wang, T. / Aronov, A.M. |
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Methods | X-ray diffraction |
Resolution | 2.69 - 2.99 Å |
Structure data | ![]() PDB-4ps3: ![]() PDB-4ps7: ![]() PDB-4ps8: |
Chemicals | ![]() ChemComp-2WH: ![]() ChemComp-HOH: ![]() ChemComp-2WJ: ![]() ChemComp-2WK: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / serine/threonine protein kinase / TRANSFERASE-TRANSFERASE INHIBITOR complex |