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-Structure paper
Title | Identification and structure-function analysis of subfamily selective g protein-coupled receptor kinase inhibitors. |
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Journal, issue, pages | Acs Chem. Biol., Vol. 10, Page 310-319, Year 2015 |
Publish date | May 23, 2014 (structure data deposition date) |
Authors | Homan, K.T. / Larimore, K.M. / Elkins, J.M. / Szklarz, M. / Knapp, S. / Tesmer, J.J. |
External links | Acs Chem. Biol. / PubMed:25238254 |
Methods | X-ray diffraction |
Resolution | 1.85 - 2.56 Å |
Structure data | PDB-4pni: PDB-4pnk: |
Chemicals | ChemComp-KQQ: ChemComp-CL: ChemComp-HOH: ChemComp-KZQ: |
Source |
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Keywords | Transferase/Transferase inhibitor / AGC FAMILY KINASE / SER/THR KINASE / RGS HOMOLOGY DOMAIN / G PROTEIN COUPLED RECEPTOR KINASE / GRK / GRK1 / RHODOPSIN KINASE / HYDROLYASE / GPCR / PHOSPHORYLATION / Transferase-Transferase inhibitor complex / PROTEIN KINASE / HYDROLASE / ATP BINDING / PERIPHERAL MEMBRANE PROTEIN |