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-Structure paper
Title | Covalent Small Molecule Inhibitors of Ca(2+)-Bound S100B. |
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Journal, issue, pages | Biochemistry, Vol. 53, Page 6628-6640, Year 2014 |
Publish date | Apr 22, 2014 (structure data deposition date) |
![]() | Cavalier, M.C. / Pierce, A.D. / Wilder, P.T. / Alasady, M.J. / Hartman, K.G. / Neau, D.B. / Foley, T.L. / Jadhav, A. / Maloney, D.J. / Simeonov, A. ...Cavalier, M.C. / Pierce, A.D. / Wilder, P.T. / Alasady, M.J. / Hartman, K.G. / Neau, D.B. / Foley, T.L. / Jadhav, A. / Maloney, D.J. / Simeonov, A. / Toth, E.A. / Weber, D.J. |
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Methods | X-ray diffraction |
Resolution | 1.08 - 2.178 Å |
Structure data | ![]() PDB-4pdz: ![]() PDB-4pe0: ![]() PDB-4pe1: ![]() PDB-4pe4: ![]() PDB-4pe7: |
Chemicals | ![]() ChemComp-CA: ![]() ChemComp-CTI: ![]() ChemComp-HOH: ![]() ChemComp-NQS: ![]() ChemComp-DCD: ![]() ChemComp-REV: ![]() ChemComp-ODN: |
Source |
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![]() | METAL BINDING PROTEIN/INHIBITOR / Malignant Melanoma / Calcium Binding / Covalent Inhibitor / Complex / METAL BINDING PROTEIN-INHIBITOR complex |