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-Structure paper
Title | Discovery of BRD4 bromodomain inhibitors by fragment-based high-throughput docking. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 24, Page 2493-2496, Year 2014 |
Publish date | Apr 15, 2014 (structure data deposition date) |
![]() | Zhao, H. / Gartenmann, L. / Dong, J. / Spiliotopoulos, D. / Caflisch, A. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.25 - 1.293 Å |
Structure data | ![]() PDB-4pce: ![]() PDB-4pci: |
Chemicals | ![]() ChemComp-EDO: ![]() ChemComp-2N0: ![]() ChemComp-HOH: ![]() ChemComp-2NJ: |
Source |
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![]() | Transcription/transcription Inhibitor / Transcription-transcription Inhibitor complex |