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-Structure paper
Title | Discovery and development of potent and selective inhibitors of histone methyltransferase g9a. |
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Journal, issue, pages | ACS Med Chem Lett, Vol. 5, Page 205-209, Year 2014 |
Publish date | Dec 5, 2013 (structure data deposition date) |
Authors | Sweis, R.F. / Pliushchev, M. / Brown, P.J. / Guo, J. / Li, F. / Maag, D. / Petros, A.M. / Soni, N.B. / Tse, C. / Vedadi, M. ...Sweis, R.F. / Pliushchev, M. / Brown, P.J. / Guo, J. / Li, F. / Maag, D. / Petros, A.M. / Soni, N.B. / Tse, C. / Vedadi, M. / Michaelides, M.R. / Chiang, G.G. / Pappano, W.N. |
External links | ACS Med Chem Lett / PubMed:24900801 |
Methods | X-ray diffraction |
Resolution | 2.03 Å |
Structure data | PDB-4nvq: |
Chemicals | ChemComp-2OD: ChemComp-SAH: ChemComp-ZN: ChemComp-HOH: |
Source |
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Keywords | Transferase/Transferase Inhibitor / Lysine Methyl Transferase / Transferase-Transferase Inhibitor complex |