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Structure paper

TitleStructure-Guided Design of Potent Diazobenzene Inhibitors for the BET Bromodomains
Journal, issue, pagesJ. Med. Chem., Vol. 56, Page 9251-9264, Year 2013
Publish dateDec 3, 2013 (structure data deposition date)
AuthorsZhang, G. / Plotnikov, A.N. / Rusinova, E. / Shen, T. / Morohashi, K. / Joshua, J. / Zeng, L. / Mujtaba, S. / Ohlmeyer, M. / Zhou, M.-M.
External linksPubMed:24144283
MethodsX-ray diffraction
Resolution1.2 - 1.4 Å
Structure data

PDB-4nuc:
Crystal structure of the first bromodomain of human BRD4 in complex with MS435 inhibitor
Method: X-RAY DIFFRACTION / Resolution: 1.4 Å

PDB-4nud:
Crystal structure of the first bromodomain of human BRD4 in complex with MS436 inhibitor
Method: X-RAY DIFFRACTION / Resolution: 1.2 Å

PDB-4nue:
Crystal structure of the first bromodomain of human BRD4 in complex with MS267 inhibitor
Method: X-RAY DIFFRACTION / Resolution: 1.3 Å

Chemicals

ChemComp-435:
4-[(E)-(4-hydroxy-3,5-dimethylphenyl)diazenyl]-N-(pyridin-2-yl)benzenesulfonamide

ChemComp-EDO:
1,2-ETHANEDIOL

ChemComp-HOH:
WATER

ChemComp-NUD:
4-[(E)-(2-amino-4-hydroxy-5-methylphenyl)diazenyl]-N-(pyridin-2-yl)benzenesulfonamide

ChemComp-NUE:
4-[(E)-(2-amino-4-hydroxy-3,5-dimethylphenyl)diazenyl]-N-(pyridin-2-yl)benzenesulfonamide

Source
  • homo sapiens (human)
KeywordsTRANSCRIPTION / Transcription factor / TRANSCRIPTION/TRANSCRIPTION INHIBITOR / TRANSCRIPTION-TRANSCRIPTION INHIBITOR complex

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