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Title | Targeting low-druggability bromodomains: fragment based screening and inhibitor design against the BAZ2B bromodomain. |
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Journal, issue, pages | J. Med. Chem., Vol. 56, Page 10183-10187, Year 2013 |
Publish date | Nov 26, 2013 (structure data deposition date) |
![]() | Ferguson, F.M. / Fedorov, O. / Chaikuad, A. / Philpott, M. / Muniz, J.R. / Felletar, I. / von Delft, F. / Heightman, T. / Knapp, S. / Abell, C. / Ciulli, A. |
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Methods | X-ray diffraction |
Resolution | 1.85 - 2.08 Å |
Structure data | ![]() PDB-4nr9: ![]() PDB-4nra: ![]() PDB-4nrb: ![]() PDB-4nrc: |
Chemicals | ![]() ChemComp-EDO: ![]() ChemComp-ALY: ![]() ChemComp-HOH: ![]() ChemComp-2LW: ![]() ChemComp-2LX: ![]() ChemComp-2LY: ![]() ChemComp-15P: |
Source |
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![]() | TRANSCRIPTION / SGC / Structural Genomics Consortium / bromodomain / acetylated lysine binding protein / KIAA1476 / WALp4 |