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-Structure paper
Title | Crystal structure of the first bromodomain of human BRD4 in complex with an isoxazolyl-benzimidazole ligand |
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Journal, issue, pages | To be Published |
Publish date | Nov 26, 2013 (structure data deposition date) |
![]() | Filippakopoulos, P. / Hay, D. / von Delft, F. / Edwards, A.M. / Picaud, S. / Fedorov, O. / Brennan, P. / Bountra, C. |
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Methods | X-ray diffraction |
Resolution | 1.635 Å |
Structure data | ![]() PDB-4nr8: |
Chemicals | ![]() ChemComp-K: ![]() ChemComp-2LL: ![]() ChemComp-EDO: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSCRIPTION/INHIBITOR / Structural Genomics Consortium / SGC / chemical tool / small molecule inhibitor / transcription / TRANSCRIPTION-INHIBITOR complex |