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-Structure paper
Title | Crystal structure of the bromodomain of human CREBBP in complex with an isoxazolyl-benzimidazole ligand |
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Journal, issue, pages | TO BE PUBLISHED |
Publish date | Nov 26, 2013 (structure data deposition date) |
![]() | Filippakopoulos, P. / Picaud, S. / Felletar, I. / Hay, D. / Fedorov, O. / Martin, S. / Krojer, T. / Nowak, R. / von Delft, F. / Brennan, P. ...Filippakopoulos, P. / Picaud, S. / Felletar, I. / Hay, D. / Fedorov, O. / Martin, S. / Krojer, T. / Nowak, R. / von Delft, F. / Brennan, P. / Arrowsmith, C.H. / Edwards, A.M. / Bountra, C. / Knapp, S. |
![]() | Search PubMed |
Methods | X-ray diffraction |
Resolution | 1.2 - 1.69 Å |
Structure data | ![]() PDB-4nr4: ![]() PDB-4nr5: ![]() PDB-4nr7: |
Chemicals | ![]() ChemComp-2LK: ![]() ChemComp-EDO: ![]() ChemComp-MG: ![]() ChemComp-HOH: ![]() ChemComp-2LL: ![]() ChemComp-NO3: ![]() ChemComp-2LO: |
Source |
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![]() | TRANSCRIPTION/INHIBITOR / Structural Genomics Consortium / SGC / chemical tool / small molecule inhibitor / transcription / TRANSCRIPTION-INHIBITOR complex / TRANSFERASE |