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-Structure paper
Title | Discovery of Tertiary Amine and Indole Derivatives as Potent ROR gamma t Inverse Agonists. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 5, Page 65-68, Year 2014 |
Publish date | Nov 6, 2013 (structure data deposition date) |
![]() | Yang, T. / Liu, Q. / Cheng, Y. / Cai, W. / Ma, Y. / Yang, L. / Wu, Q. / Orband-Miller, L.A. / Zhou, L. / Xiang, Z. ...Yang, T. / Liu, Q. / Cheng, Y. / Cai, W. / Ma, Y. / Yang, L. / Wu, Q. / Orband-Miller, L.A. / Zhou, L. / Xiang, Z. / Huxdorf, M. / Zhang, W. / Zhang, J. / Xiang, J.N. / Leung, S. / Qiu, Y. / Zhong, Z. / Elliott, J.D. / Lin, X. / Wang, Y. |
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Methods | X-ray diffraction |
Resolution | 2.01 Å |
Structure data | ![]() PDB-4nie: |
Chemicals | ![]() ChemComp-NBH: ![]() ChemComp-DMX: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSCRIPTION/AGONIST / nuclear receptor / ligand binding domain / TRANSCRIPTION-AGONIST complex |