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Title | Glucocorticoid receptor modulators informed by crystallography lead to a new rationale for receptor selectivity, function, and implications for structure-based design. |
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Journal, issue, pages | J. Med. Chem., Vol. 57, Page 849-860, Year 2014 |
Publish date | Jul 22, 2013 (structure data deposition date) |
![]() | Carson, M.W. / Luz, J.G. / Suen, C. / Montrose, C. / Zink, R. / Ruan, X. / Cheng, C. / Cole, H. / Adrian, M.D. / Kohlman, D.T. ...Carson, M.W. / Luz, J.G. / Suen, C. / Montrose, C. / Zink, R. / Ruan, X. / Cheng, C. / Cole, H. / Adrian, M.D. / Kohlman, D.T. / Mabry, T. / Snyder, N. / Condon, B. / Maletic, M. / Clawson, D. / Pustilnik, A. / Coghlan, M.J. |
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Methods | X-ray diffraction |
Resolution | 2.35 Å |
Structure data | ![]() PDB-4lsj: |
Chemicals | ![]() ChemComp-LSJ: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSCRIPTION / nuclear hormone receptor |