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-Structure paper
Title | Crystal Structures of PI3K alpha Complexed with PI103 and Its Derivatives: New Directions for Inhibitors Design. |
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Journal, issue, pages | ACS Med Chem Lett, Vol. 5, Page 138-142, Year 2014 |
Publish date | Jun 3, 2013 (structure data deposition date) |
Authors | Zhao, Y. / Zhang, X. / Chen, Y. / Lu, S. / Peng, Y. / Wang, X. / Guo, C. / Zhou, A. / Zhang, J. / Luo, Y. ...Zhao, Y. / Zhang, X. / Chen, Y. / Lu, S. / Peng, Y. / Wang, X. / Guo, C. / Zhou, A. / Zhang, J. / Luo, Y. / Shen, Q. / Ding, J. / Meng, L. |
External links | ACS Med Chem Lett / PubMed:24900786 |
Methods | X-ray diffraction |
Resolution | 2.501 - 2.8 Å |
Structure data | PDB-4l1b: PDB-4l23: PDB-4l2y: |
Chemicals | ChemComp-SO4: ChemComp-HOH: ChemComp-X6K: ChemComp-GOL: ChemComp-XXK: |
Source |
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Keywords | signaling Protein/transferase/Inhibitor / ATP binding / signaling Protein-transferase-Inhibitor complex / PI-103 |