+Search query
-Structure paper
Title | Structure-Efficiency Relationship of [1,2,4]Triazol-3-ylamines as Novel Nicotinamide Isosteres that Inhibit Tankyrases. |
---|---|
Journal, issue, pages | J. Med. Chem., Vol. 56, Page 7049-7059, Year 2013 |
Publish date | May 17, 2013 (structure data deposition date) |
Authors | Shultz, M.D. / Majumdar, D. / Chin, D.N. / Fortin, P.D. / Feng, Y. / Gould, T. / Kirby, C.A. / Stams, T. / Waters, N.J. / Shao, W. |
External links | J. Med. Chem. / PubMed:23879431 |
Methods | X-ray diffraction |
Resolution | 2.29 Å |
Structure data | PDB-4krs: |
Chemicals | ChemComp-ZN: ChemComp-SO4: ChemComp-1SX: ChemComp-HOH: |
Source |
|
Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / TRANSFERASE-TRANSFERASE INHIBITOR complex |