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-Structure paper
Title | Extension into the entrance channel of HIV-1 reverse transcriptase-Crystallography and enhanced solubility. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 23, Page 5209-5212, Year 2013 |
Publish date | May 6, 2013 (structure data deposition date) |
![]() | Bollini, M. / Frey, K.M. / Cisneros, J.A. / Spasov, K.A. / Das, K. / Bauman, J.D. / Arnold, E. / Anderson, K.S. / Jorgensen, W.L. |
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Methods | X-ray diffraction |
Resolution | 1.95 - 2.89 Å |
Structure data | ![]() PDB-4kko: ![]() PDB-4ko0: |
Chemicals | ![]() ChemComp-1RE: ![]() ChemComp-JLJ: ![]() ChemComp-SO4: ![]() ChemComp-EDO: ![]() ChemComp-HOH: |
Source |
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![]() | HYDROLASE/HYDROLASE INHIBITOR / Polymerase / Transferase / Hydrolase/inhibitor / Rnase / HYDROLASE-HYDROLASE INHIBITOR complex / P51/P66 / HETERO DIMER / NNRTI / NONNUCLEOSIDE INHIBITOR / AIDS / HIV / DNA RECOMBINATION / RNA-DIRECTED DNA POLYMERASE / DNA POLYMERASE / ENDONUCLEASE / HYDROLASE / MULTIFUNCTIONAL ENZYME / HYDROLASE-INHIBITOR COMPLEX |