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-Structure paper
Title | Structure-based identification of ureas as novel nicotinamide phosphoribosyltransferase (nampt) inhibitors. |
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Journal, issue, pages | J. Med. Chem., Vol. 56, Page 4921-4937, Year 2013 |
Publish date | Mar 21, 2013 (structure data deposition date) |
![]() | Zheng, X. / Bauer, P. / Baumeister, T. / Buckmelter, A.J. / Caligiuri, M. / Clodfelter, K.H. / Han, B. / Ho, Y.C. / Kley, N. / Lin, J. ...Zheng, X. / Bauer, P. / Baumeister, T. / Buckmelter, A.J. / Caligiuri, M. / Clodfelter, K.H. / Han, B. / Ho, Y.C. / Kley, N. / Lin, J. / Reynolds, D.J. / Sharma, G. / Smith, C.C. / Wang, Z. / Dragovich, P.S. / Oh, A. / Wang, W. / Zak, M. / Gunzner-Toste, J. / Zhao, G. / Yuen, P.W. / Bair, K.W. |
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Methods | X-ray diffraction |
Resolution | 1.6 - 1.906 Å |
Structure data | ![]() PDB-4jr5: ![]() PDB-4kfn: ![]() PDB-4kfo: |
Chemicals | ![]() ChemComp-1LS: ![]() ChemComp-PO4: ![]() ChemComp-EDO: ![]() ChemComp-HOH: ![]() ChemComp-1QR: ![]() ChemComp-1QS: |
Source |
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![]() | Transferase/Transferase inhibitor / Transferase-Transferase inhibitor complex |