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-Structure paper
Title | Azaindole-Based Inhibitors of Cdc7 Kinase: Impact of the Pre-DFG Residue, Val 195. |
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Journal, issue, pages | ACS Med Chem Lett, Vol. 4, Page 211-215, Year 2013 |
Publish date | Jan 10, 2013 (structure data deposition date) |
![]() | Tong, Y. / Stewart, K.D. / Florjancic, A.S. / Harlan, J.E. / Merta, P.J. / Przytulinska, M. / Soni, N. / Swinger, K.K. / Zhu, H. / Johnson, E.F. ...Tong, Y. / Stewart, K.D. / Florjancic, A.S. / Harlan, J.E. / Merta, P.J. / Przytulinska, M. / Soni, N. / Swinger, K.K. / Zhu, H. / Johnson, E.F. / Shoemaker, A.R. / Penning, T.D. |
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Methods | X-ray diffraction |
Resolution | 3.12 Å |
Structure data | ![]() PDB-4iq6: |
Chemicals | ![]() ChemComp-IQ6: |
Source |
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![]() | Transferase/Transferase Inhibitor / protein kinase / Transferase-Transferase Inhibitor complex |