+Search query
-Structure paper
Title | Inhibiting NF-KB-inducing kinase (NIK): Discovery, structure-based design, synthesis, structure activity relationship, and co-crystal structures |
---|---|
Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 23, Page 1238-1244, Year 2013 |
Publish date | Dec 13, 2012 (structure data deposition date) |
![]() | Li, K. / McGee, L.R. / Fisher, B. / Sudom, A. / Liu, J. / Rubenstein, S.M. / Anwer, M.K. / Cushing, T.D. / Shin, Y. / Ayres, M. ...Li, K. / McGee, L.R. / Fisher, B. / Sudom, A. / Liu, J. / Rubenstein, S.M. / Anwer, M.K. / Cushing, T.D. / Shin, Y. / Ayres, M. / Lee, F. / Eksterowicz, J. / Faulder, P. / Waszkowycz, B. / Plotnikova, O. / Farrelly, E. / Xiao, S.H. / Chen, G. / Wang, Z. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.4 - 2.9 Å |
Structure data | ![]() PDB-4idt: ![]() PDB-4idv: |
Chemicals | ![]() ChemComp-T28: ![]() ChemComp-HOH: ![]() ChemComp-13V: |
Source |
|
![]() | Transferase/Transferase Inhibitor / NIK / Nuclear factor (NF)-kB / p100 processing / 2-aminopyrimidine / Transferase-Transferase Inhibitor complex |