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-Structure paper
Title | Structure-Based Design of High-Affinity Macrocyclic Peptidomimetics to Block the Menin-Mixed Lineage Leukemia 1 (MLL1) Protein-Protein Interaction. |
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Journal, issue, pages | J. Med. Chem., Vol. 56, Page 1113-1123, Year 2013 |
Publish date | Dec 1, 2012 (structure data deposition date) |
![]() | Zhou, H. / Liu, L. / Huang, J. / Bernard, D. / Karatas, H. / Navarro, A. / Lei, M. / Wang, S. |
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Methods | X-ray diffraction |
Resolution | 3.1 Å |
Structure data | ![]() PDB-4i80: |
Source |
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![]() | TRANSCRIPTION/INHIBITOR / menin / MEN1 / MLL / macrocyclic peptidomimetic / TRANSCRIPTION / TRANSCRIPTION-INHIBITOR complex |