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-Structure paper
Title | Structure-Based Design of Potent and Selective CK1 gamma Inhibitors. |
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Journal, issue, pages | ACS Med Chem Lett, Vol. 3, Page 1059-1064, Year 2012 |
Publish date | Oct 8, 2012 (structure data deposition date) |
Authors | Huang, H. / Acquaviva, L. / Berry, V. / Bregman, H. / Chakka, N. / O'Connor, A. / DiMauro, E.F. / Dovey, J. / Epstein, O. / Grubinska, B. ...Huang, H. / Acquaviva, L. / Berry, V. / Bregman, H. / Chakka, N. / O'Connor, A. / DiMauro, E.F. / Dovey, J. / Epstein, O. / Grubinska, B. / Goldstein, J. / Gunaydin, H. / Hua, Z. / Huang, X. / Huang, L. / Human, J. / Long, A. / Newcomb, J. / Patel, V.F. / Saffran, D. / Serafino, R. / Schneider, S. / Strathdee, C. / Tang, J. / Turci, S. / White, R. / Yu, V. / Zhao, H. / Wilson, C. / Martin, M.W. |
External links | ACS Med Chem Lett / PubMed:24900428 |
Methods | X-ray diffraction |
Resolution | 1.8 - 2.4 Å |
Structure data | PDB-4hgl: PDB-4hgt: |
Chemicals | ChemComp-0YO: ChemComp-SO4: ChemComp-HOH: ChemComp-15G: |
Source |
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Keywords | transferase/transferase inhibitor / ck1g / kinase / inhibitor / transferase-transferase inhibitor complex / ck1d |