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-Structure paper
Title | Mechanism and In Vitro Pharmacology of TAK1 Inhibition by (5Z)-7-Oxozeaenol. |
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Journal, issue, pages | Acs Chem. Biol., Vol. 8, Page 643-650, Year 2013 |
Publish date | Aug 27, 2012 (structure data deposition date) |
Authors | Wu, J. / Powell, F. / Larsen, N.A. / Lai, Z. / Byth, K.F. / Read, J. / Gu, R.F. / Roth, M. / Toader, D. / Saeh, J.C. / Chen, H. |
External links | Acs Chem. Biol. / PubMed:23272696 |
Methods | X-ray diffraction |
Resolution | 2.2 Å |
Structure data | PDB-4gs6: |
Chemicals | ChemComp-EDO: ChemComp-1FM: ChemComp-HOH: |
Source |
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Keywords | Transferase/Transferase inhibitor / Kinase Fold / Tab1 binding / Cytosol / Transferase-Transferase inhibitor complex |