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Title | Optimization of Inhibitors of the Tyrosine Kinase EphB4. 2. Cellular Potency Improvement and Binding Mode Validation by X-ray Crystallography. |
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Journal, issue, pages | J. Med. Chem., Vol. 56, Page 84-96, Year 2013 |
Publish date | Aug 10, 2012 (structure data deposition date) |
![]() | Lafleur, K. / Dong, J. / Huang, D. / Caflisch, A. / Nevado, C. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.898 - 2.195 Å |
Structure data | ![]() PDB-4gk2: ![]() PDB-4gk3: ![]() PDB-4gk4: |
Chemicals | ![]() ChemComp-L66: ![]() ChemComp-HOH: ![]() ChemComp-L87: ![]() ChemComp-L90: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / RECEPTOR TYROSINE KINASE / ATP-BINDING / PHOSPHORYLATION / MEMBRANE / TRANSFERASE-TRANSFERASE INHIBITOR complex |