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-Structure paper
Title | Discovery of a novel chemotype of tyrosine kinase inhibitors by fragment-based docking and molecular dynamics. |
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Journal, issue, pages | ACS MED. CHEM. LETT., Vol. 3, Page 834-838, Year 2012 |
Publish date | Jul 12, 2012 (structure data deposition date) |
![]() | Zhao, H. / Dong, J. / Lafleur, K. / Nevado, C. / Caflisch, A. |
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Methods | X-ray diffraction |
Resolution | 1.699 Å |
Structure data | ![]() PDB-4g2f: |
Chemicals | ![]() ChemComp-C07: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / RECEPTOR TYROSINE KINASE / ATP Binding / Phosphorylation / Membrane / TRANSFERASE-TRANSFERASE INHIBITOR complex |