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-Structure paper
Title | Small molecule regulation of protein conformation by binding in the Flap of HIV protease. |
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Journal, issue, pages | Acs Chem. Biol., Vol. 8, Page 1223-1231, Year 2013 |
Publish date | Apr 6, 2012 (structure data deposition date) |
![]() | Tiefenbrunn, T. / Forli, S. / Baksh, M.M. / Chang, M.W. / Happer, M. / Lin, Y.C. / Perryman, A.L. / Rhee, J.K. / Torbett, B.E. / Olson, A.J. ...Tiefenbrunn, T. / Forli, S. / Baksh, M.M. / Chang, M.W. / Happer, M. / Lin, Y.C. / Perryman, A.L. / Rhee, J.K. / Torbett, B.E. / Olson, A.J. / Elder, J.H. / Finn, M.G. / Stout, C.D. |
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Methods | X-ray diffraction |
Resolution | 1.103 - 2.445 Å |
Structure data | ![]() PDB-4ej8: ![]() PDB-4ejd: ![]() PDB-4ejk: ![]() PDB-4ejl: |
Chemicals | ![]() ChemComp-DMS: ![]() ChemComp-EDO: ![]() ChemComp-1F1: ![]() ChemComp-HOH: ![]() ChemComp-BME: ![]() ChemComp-GOL: ![]() ChemComp-IOP: ![]() ChemComp-PEG: |
Source |
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![]() | HYDROLASE / apo protease / allostery / fragment binding / closed form / HYDROLASE/HYDROLASE INHIBITOR / HYDROLASE-HYDROLASE INHIBITOR complex |