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-Structure paper
Title | Small molecule regulation of protein conformation by binding in the Flap of HIV protease. |
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Journal, issue, pages | Acs Chem. Biol., Vol. 8, Page 1223-1231, Year 2013 |
Publish date | Apr 6, 2012 (structure data deposition date) |
Authors | Tiefenbrunn, T. / Forli, S. / Baksh, M.M. / Chang, M.W. / Happer, M. / Lin, Y.C. / Perryman, A.L. / Rhee, J.K. / Torbett, B.E. / Olson, A.J. ...Tiefenbrunn, T. / Forli, S. / Baksh, M.M. / Chang, M.W. / Happer, M. / Lin, Y.C. / Perryman, A.L. / Rhee, J.K. / Torbett, B.E. / Olson, A.J. / Elder, J.H. / Finn, M.G. / Stout, C.D. |
External links | Acs Chem. Biol. / PubMed:23540839 |
Methods | X-ray diffraction |
Resolution | 1.103 - 2.445 Å |
Structure data | PDB-4ej8: PDB-4ejd: PDB-4ejk: PDB-4ejl: |
Chemicals | ChemComp-DMS: ChemComp-EDO: ChemComp-1F1: ChemComp-HOH: ChemComp-BME: ChemComp-GOL: ChemComp-IOP: ChemComp-PEG: |
Source |
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Keywords | HYDROLASE / apo protease / allostery / fragment binding / closed form / HYDROLASE/HYDROLASE INHIBITOR / HYDROLASE-HYDROLASE INHIBITOR complex |