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-Structure paper
Title | Discovery and characterization of novel allosteric FAK inhibitors. |
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Journal, issue, pages | Eur. J. Med. Chem., Vol. 61, Page 49-60, Year 2013 |
Publish date | Mar 25, 2012 (structure data deposition date) |
Authors | Iwatani, M. / Iwata, H. / Okabe, A. / Skene, R.J. / Tomita, N. / Hayashi, Y. / Aramaki, Y. / Hosfield, D.J. / Hori, A. / Baba, A. / Miki, H. |
External links | Eur. J. Med. Chem. / PubMed:22819505 |
Methods | X-ray diffraction |
Resolution | 1.67 - 2.65 Å |
Structure data | PDB-4ebv: PDB-4ebw: |
Chemicals | ChemComp-0O7: ChemComp-IPA: ChemComp-HOH: ChemComp-0PF: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / Kinase Domain / Allosteric inhibitor / TRANSFERASE-TRANSFERASE INHIBITOR complex |