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-Structure paper
Title | Reversible targeting of noncatalytic cysteines with chemically tuned electrophiles. |
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Journal, issue, pages | Nat. Chem. Biol., Vol. 8, Page 471-476, Year 2012 |
Publish date | Jan 12, 2012 (structure data deposition date) |
Authors | Serafimova, I.M. / Pufall, M.A. / Krishnan, S. / Duda, K. / Cohen, M.S. / Maglathlin, R.L. / McFarland, J.M. / Miller, R.M. / Frodin, M. / Taunton, J. |
External links | Nat. Chem. Biol. / PubMed:22466421 |
Methods | X-ray diffraction |
Resolution | 2.4 Å |
Structure data | PDB-4d9t: PDB-4d9u: |
Chemicals | ChemComp-0JG: ChemComp-NA: ChemComp-HOH: ChemComp-0JH: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / kinase / inhibitor / reversible / thiol / phosphorylation / migration / TRANSFERASE-TRANSFERASE INHIBITOR complex / reversible inhibitor |