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-Structure paper
Title | Plasmepsin Inhibitory Activity and Structure-Guided Optimization of a Potent Hydroxyethylamine-Based Antimalarial Hit. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 5, Page 373-, Year 2014 |
Publish date | Jan 8, 2014 (structure data deposition date) |
Authors | Jaudzems, K. / Tars, K. / Maurops, G. / Ivdra, N. / Otikovs, M. / Leitans, J. / Kanepe-Lapsa, I. / Domraceva, I. / Mutule, I. / Trapencieris, P. ...Jaudzems, K. / Tars, K. / Maurops, G. / Ivdra, N. / Otikovs, M. / Leitans, J. / Kanepe-Lapsa, I. / Domraceva, I. / Mutule, I. / Trapencieris, P. / Blackman, M.J. / Jirgensons, A. |
External links | Acs Med. Chem. Lett. / PubMed:24900843 |
Methods | X-ray diffraction |
Resolution | 1.85 Å |
Structure data | PDB-4cku: |
Chemicals | ChemComp-P2F: ChemComp-HOH: |
Source |
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Keywords | HYDROLASE / MALARIA / DRUG DESIGN |