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-Structure paper
Title | The Commonly Used Pi3-Kinase Probe Ly294002 is an Inhibitor of Bet Bromodomains. |
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Journal, issue, pages | Acs Chem. Biol., Vol. 9, Page 495-, Year 2014 |
Publish date | Nov 18, 2013 (structure data deposition date) |
Authors | Dittmann, A. / Werner, T. / Chung, C. / Savitski, M.M. / Falth Savitski, M. / Grandi, P. / Hopf, C. / Lindon, M. / Neubauer, G. / Prinjha, R.K. ...Dittmann, A. / Werner, T. / Chung, C. / Savitski, M.M. / Falth Savitski, M. / Grandi, P. / Hopf, C. / Lindon, M. / Neubauer, G. / Prinjha, R.K. / Bantscheff, M. / Drewes, G. |
External links | Acs Chem. Biol. / PubMed:24533473 |
Methods | X-ray diffraction |
Resolution | 1.32 - 1.55 Å |
Structure data | PDB-4cfk: PDB-4cfl: |
Chemicals | ChemComp-GOL: ChemComp-LY2: ChemComp-EDO: ChemComp-HOH: ChemComp-8DQ: |
Source |
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Keywords | CELL CYCLE / INHIBITOR / HISTONE / EPIGENETIC READER / ANTAGONIST / KINASE |