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-Structure paper
| Title | Bisubstrate Udp-Peptide Conjugates as Human O-Glcnac Transferase Inhibitors. |
|---|---|
| Journal, issue, pages | Biochem. J., Vol. 457, Page 497-, Year 2014 |
| Publish date | Nov 5, 2013 (structure data deposition date) |
Authors | Borodkin, V.S. / Schimpl, M. / Gundogdu, M. / Rafie, K. / Dorfmueller, H.C. / Robinson, D.A. / Van Aalten, D.M. |
External links | Biochem. J. / PubMed:24256146 |
| Methods | X-ray diffraction |
| Resolution | 3.15 Å |
| Structure data | ![]() PDB-4cdr: |
| Chemicals | ![]() ChemComp-SO4: ![]() ChemComp-UDP: |
| Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX / INVERTING GT-B ENZYME / BI-SUBSTRATE ANALOG INHIBITOR |
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homo sapiens (human)
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