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-Structure paper
Title | Discovery of Pyrroloaminopyrazoles as Novel Pak Inhibitors. |
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Journal, issue, pages | J. Med. Chem., Vol. 55, Page 4728-, Year 2012 |
Publish date | Apr 4, 2012 (structure data deposition date) |
![]() | Guo, C. / Mcalpine, I. / Zhang, J. / Knighton, D.D. / Kephart, S. / Johnson, M.C. / Li, H. / Bouzida, D. / Yang, A. / Dong, L. ...Guo, C. / Mcalpine, I. / Zhang, J. / Knighton, D.D. / Kephart, S. / Johnson, M.C. / Li, H. / Bouzida, D. / Yang, A. / Dong, L. / Marakovits, J. / Tikhe, J. / Richardson, P. / Guo, L.C. / Kania, R. / Edwards, M.P. / Kraynov, E. / Christensen, J. / Piraino, J. / Lee, J. / Dagostino, E. / Del-Carmen, C. / Deng, Y.L. / Smeal, T. / Murray, B.W. |
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Methods | X-ray diffraction |
Resolution | 2.2 Å |
Structure data | ![]() PDB-4app: |
Chemicals | ![]() ChemComp-N53: ![]() ChemComp-GOL: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE / PROTEIN KINASE |