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-Structure paper
Title | Inhibition of Leishmania Infantum Trypanothione Reductase by Azole-Based Compounds: A Comparative Analysis with its Physiological Substrate by X-Ray Crystallography. |
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Journal, issue, pages | Chemmedchem, Vol. 8, Page 1175-, Year 2013 |
Publish date | Jan 4, 2012 (structure data deposition date) |
![]() | Baiocco, P. / Poce, G. / Alfonso, S. / Cocozza, M. / Porretta, G.C. / Colotti, G. / Biava, M. / Moraca, F. / Botta, M. / Yardley, V. ...Baiocco, P. / Poce, G. / Alfonso, S. / Cocozza, M. / Porretta, G.C. / Colotti, G. / Biava, M. / Moraca, F. / Botta, M. / Yardley, V. / Fiorillo, A. / Lantella, A. / Malatesta, F. / Ilari, A. |
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Methods | X-ray diffraction |
Resolution | 3.2 - 3.61 Å |
Structure data | ![]() PDB-4adw: ![]() PDB-4apn: |
Chemicals | ![]() ChemComp-FAD: ![]() ChemComp-NDP: ![]() ChemComp-GCG: ![]() ChemComp-JV0: ![]() ChemComp-HOH: |
Source |
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![]() | OXIDOREDUCTASE / INHIBITION MECHANISM / TRYPANOSOMATIDS |