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-Structure paper
Title | Inhibitors of Acetyltransferase Domain of N-Acetylglucosamine-1-Phosphate-Uridyltransferase/ Glucosamine-1-Phosphate-Acetyltransferase (Glmu). Part 1: Hit to Lead Evaluation of a Novel Arylsulfonamide Series. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 22, Page 1510-, Year 2012 |
Publish date | Nov 30, 2011 (structure data deposition date) |
![]() | Green, O.M. / McKenzie, A.R. / Shapiro, A.B. / Otterbein, L. / Ni, H. / Patten, A. / Stokes, S. / Albert, R. / Kawatkar, S. / Breed, J. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2 - 2.2 Å |
Structure data | ![]() PDB-4aa7: ![]() PDB-4aaw: ![]() PDB-4ac3: |
Chemicals | ![]() ChemComp-R82: ![]() ChemComp-SO4: ![]() ChemComp-HOH: ![]() ChemComp-R84: ![]() ChemComp-R83: |
Source |
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![]() | TRANSFERASE / ACETYL TRANSFERASE / TRANSFERASE-INHIBITOR COMPLEX / TRANSFERASE INHIBITOR COMPLEX |