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-Structure paper
Title | Hit to Lead Evaluation of 1,2,3-Triazolo[4,5-B]Pyridines as Pim Kinase Inhibitors. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 22, Page 1591-, Year 2012 |
Publish date | Nov 12, 2011 (structure data deposition date) |
![]() | Pastor, J. / Oyarzabal, J. / Saluste, G. / Alvarez, R.M. / Rivero, V. / Ramos, F. / Cendon, E. / Blanco-Aparicio, C. / Ajenjo, N. / Cebria, A. ...Pastor, J. / Oyarzabal, J. / Saluste, G. / Alvarez, R.M. / Rivero, V. / Ramos, F. / Cendon, E. / Blanco-Aparicio, C. / Ajenjo, N. / Cebria, A. / Albarran, M.I. / Cebrian, D. / Corrionero, A. / Fominaya, J. / Montoya, G. / Mazzorana, M. |
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Methods | X-ray diffraction |
Resolution | 2.3 Å |
Structure data | ![]() PDB-4a7c: |
Chemicals | ![]() ChemComp-E46: ![]() ChemComp-IMD: ![]() ChemComp-ACT: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE / PROTEIN KINASE / INHIBITOR |