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-Structure paper
Title | Diaminopyridine-based potent and selective mps1 kinase inhibitors binding to an unusual flipped-Peptide conformation. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 3, Page 560-564, Year 2012 |
Publish date | Mar 30, 2012 (structure data deposition date) |
![]() | Kusakabe, K. / Ide, N. / Daigo, Y. / Itoh, T. / Higashino, K. / Okano, Y. / Tadano, G. / Tachibana, Y. / Sato, Y. / Inoue, M. ...Kusakabe, K. / Ide, N. / Daigo, Y. / Itoh, T. / Higashino, K. / Okano, Y. / Tadano, G. / Tachibana, Y. / Sato, Y. / Inoue, M. / Wada, T. / Iguchi, M. / Kanazawa, T. / Ishioka, Y. / Dohi, K. / Tagashira, S. / Kido, Y. / Sakamoto, S. / Yasuo, K. / Maeda, M. / Yamamoto, T. / Higaki, M. / Endoh, T. / Ueda, K. / Shiota, T. / Murai, H. / Nakamura, Y. |
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Methods | X-ray diffraction |
Resolution | 2.4 Å |
Structure data | ![]() PDB-3vqu: |
Chemicals | ![]() ChemComp-IOD: ![]() ChemComp-O22: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / KINASE / SERINE/THREONINE-PROTEIN KINASE / TRANSFERASE-TRANSFERASE INHIBITOR complex |