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-Structure paper
Title | Discovery of potent and selective covalent inhibitors of JNK. |
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Journal, issue, pages | Chem. Biol., Vol. 19, Page 140-154, Year 2012 |
Publish date | Dec 20, 2011 (structure data deposition date) |
![]() | Zhang, T. / Inesta-Vaquera, F. / Niepel, M. / Zhang, J. / Ficarro, S.B. / Machleidt, T. / Xie, T. / Marto, J.A. / Kim, N. / Sim, T. ...Zhang, T. / Inesta-Vaquera, F. / Niepel, M. / Zhang, J. / Ficarro, S.B. / Machleidt, T. / Xie, T. / Marto, J.A. / Kim, N. / Sim, T. / Laughlin, J.D. / Park, H. / LoGrasso, P.V. / Patricelli, M. / Nomanbhoy, T.K. / Sorger, P.K. / Alessi, D.R. / Gray, N.S. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.6 - 2.97 Å |
Structure data | ![]() PDB-3v6r: ![]() PDB-3v6s: |
Chemicals | ![]() ChemComp-CQQ: ![]() ChemComp-HOH: ![]() ChemComp-0F0: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / KINASE FOLD / APOPTOSIS / MAP KINASE / CYS modification / Phosphorylation / JNK / TRANSFERASE-TRANSFERASE INHIBITOR complex |