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-Structure paper
Title | Targeting the Hinge Glycine Flip and the Activation Loop: Novel Approach to Potent p38 alpha Inhibitors. |
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Journal, issue, pages | J. Med. Chem., Vol. 55, Page 7862-7874, Year 2012 |
Publish date | Nov 30, 2011 (structure data deposition date) |
![]() | Martz, K.E. / Dorn, A. / Baur, B. / Schattel, V. / Goettert, M.I. / Mayer-Wrangowski, S.C. / Rauh, D. / Laufer, S.A. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.4 Å |
Structure data | ![]() PDB-3uvp: |
Chemicals | ![]() ChemComp-048: ![]() ChemComp-BOG: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / protein kinase / selective p38 inhibitor / SAR / benzosuberon derivative / TRANSFERASE-TRANSFERASE INHIBITOR complex |