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-Structure paper
Title | Structural basis of selective inhibition of human tankyrases. |
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Journal, issue, pages | J. Med. Chem., Vol. 55, Page 1360-1367, Year 2012 |
Publish date | Oct 19, 2011 (structure data deposition date) |
Authors | Narwal, M. / Venkannagari, H. / Lehtio, L. |
External links | J. Med. Chem. / PubMed:22233320 |
Methods | X-ray diffraction |
Resolution | 1.75 - 2.3 Å |
Structure data | PDB-3u9h: PDB-3u9y: PDB-3ua9: |
Chemicals | ChemComp-ZN: ChemComp-SO4: ChemComp-NCA: ChemComp-GOL: ChemComp-PEG: ChemComp-HOH: ChemComp-09L: ChemComp-IWR: |
Source |
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Keywords | TRANSFERASE / PROTEIN-LIGAND COMPLEX / DIPHTHERIA TOXIN LIKE FOLD / ADP-RIBOSYLATION / TRANSFERASE/TRANSFERASE INHIBITOR / TRANSFERASE-TRANSFERASE INHIBITOR complex |