+Search query
-Structure paper
Title | Highly specific, bisubstrate-competitive Src inhibitors from DNA-templated macrocycles. |
---|---|
Journal, issue, pages | Nat. Chem. Biol., Vol. 8, Page 366-374, Year 2012 |
Publish date | Oct 10, 2011 (structure data deposition date) |
Authors | Georghiou, G. / Kleiner, R.E. / Pulkoski-Gross, M. / Liu, D.R. / Seeliger, M.A. |
External links | Nat. Chem. Biol. / PubMed:22344177 |
Methods | X-ray diffraction |
Resolution | 1.9 - 2.241 Å |
Structure data | PDB-3u4w: PDB-3u51: |
Chemicals | ChemComp-GOL: ChemComp-SO4: ChemComp-HOH: |
Source |
|
Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / protein kinase / Src-like inactive conformation / TRANSFERASE-TRANSFERASE INHIBITOR complex |