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-Structure paper
Title | A novel compound from a molecular fragment library screen inhibits glycosyltransferases by displacing the metal ion and interfering with substrate binding |
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Journal, issue, pages | To be Published |
Publish date | Sep 29, 2011 (structure data deposition date) |
![]() | Jorgensen, R. / Grimm, L.L. / Sindhuwinata, N. / Peters, T. / Palcic, M.M. |
![]() | Search PubMed |
Methods | X-ray diffraction |
Resolution | 1.6 - 1.85 Å |
Structure data | ![]() PDB-3u0x: ![]() PDB-3u0y: |
Chemicals | ![]() ChemComp-GTI: ![]() ChemComp-CL: ![]() ChemComp-GOL: ![]() ChemComp-SO4: ![]() ChemComp-HOH: ![]() ChemComp-UDP: ![]() ChemComp-MN: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / ROSSMANN FOLD / OPEN CONFORMATION / GLYCOSYLTRANSFERASE / TRANSFERASE GTB / ABO / BLOOD GROUP ANTIGEN / GLYCOPROTEIN / METAL-BINDING / MANGANESE / UDP-GAL / H-ANTIGEN ACCEPTOR / MEMBRANE / TRANSFERASE-TRANSFERASE INHIBITOR complex / "SEMI CLOSED" CONFORMATION / transferase |