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Title | Fragment-Based Screening for Inhibitors of PDE4A Using Enthalpy Arrays and X-ray Crystallography. |
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Journal, issue, pages | J Biomol Screen, Vol. 17, Page 469-480, Year 2012 |
Publish date | Sep 20, 2011 (structure data deposition date) |
Authors | Recht, M.I. / Sridhar, V. / Badger, J. / Hernandez, L. / Chie-Leon, B. / Nienaber, V. / Torres, F.E. |
External links | J Biomol Screen / PubMed:22223051 |
Methods | X-ray diffraction |
Resolution | 2.84 Å |
Structure data | PDB-3tvx: |
Chemicals | ChemComp-ZN: ChemComp-MG: ChemComp-PNX: ChemComp-SO4: |
Source |
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Keywords | HYDROLASE/HYDROLASE INHIBITOR / HYDROLASE / HYDROLASE-HYDROLASE INHIBITOR complex |