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-Structure paper
Title | Flexibility of the flap in the active site of BACE1 as revealed by crystal structures and molecular dynamics simulations |
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Journal, issue, pages | Acta Crystallogr. ,Sect. D, Vol. 68, Page 13-25, Year 2012 |
Publish date | Sep 8, 2011 (structure data deposition date) |
![]() | Xu, Y.C. / Li, M.J. / Greenblatt, H. / Chen, W.Y. / Paz, A. / Dym, O. / Peleg, Y. / Chen, T.T. / Shen, X. / He, J.H. ...Xu, Y.C. / Li, M.J. / Greenblatt, H. / Chen, W.Y. / Paz, A. / Dym, O. / Peleg, Y. / Chen, T.T. / Shen, X. / He, J.H. / Jiang, H.L. / Silman, I. / Sussman, J.L. |
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Methods | X-ray diffraction |
Resolution | 1.6 - 2.55 Å |
Structure data | ![]() PDB-3tpj: ![]() PDB-3tpl: ![]() PDB-3tpp: ![]() PDB-3tpr: |
Chemicals | ![]() ChemComp-SO4: ![]() ChemComp-CL: ![]() ChemComp-URE: ![]() ChemComp-HOH: ![]() ChemComp-5HA: |
Source |
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![]() | HYDROLASE / PROTEASE / MEMAPSIN 2 / BACE1 / Beta-secretase 1 / HYDROLASE/HYDROLASE INHIBITOR / HYDROLASE-HYDROLASE INHIBITOR complex |