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| Title | Structure-Guided Design of a High-Affinity Platelet Integrin alphaIIbbeta3 Receptor Antagonist That Disrupts Mg2+ Binding to the MIDAS |
|---|---|
| Journal, issue, pages | Sci Transl Med, Vol. 4, Page 125ra32-125ra32, Year 2012 |
| Publish date | Jul 25, 2011 (structure data deposition date) |
Authors | Zhu, J. / Choi, W.S. / McCoy, J.G. / Negri, A. / Naini, S. / Li, J. / Shen, M. / Huang, W. / Bougie, D. / Rasmussen, M. ...Zhu, J. / Choi, W.S. / McCoy, J.G. / Negri, A. / Naini, S. / Li, J. / Shen, M. / Huang, W. / Bougie, D. / Rasmussen, M. / Aster, R. / Thomas, C.J. / Filizola, M. / Springer, T.A. / Coller, B.S. |
External links | Sci Transl Med / PubMed:22422993 |
| Methods | X-ray diffraction |
| Resolution | 2.2 - 2.6 Å |
| Structure data | ![]() PDB-3t3m: ![]() PDB-3t3p: |
| Chemicals | ![]() ChemComp-CA: ![]() ChemComp-RC2: ![]() ChemComp-SO4: ![]() ChemComp-NAG: ![]() ChemComp-CL: ![]() ChemComp-HOH: ![]() ChemComp-GOL: ![]() ChemComp-MG: |
| Source |
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Keywords | CELL ADHESION / integrin / blood clotting / Fibrinogen / platelet |
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