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-Structure paper
Title | Selective Inhibitors of Histone Methyltransferase DOT1L: Design, Synthesis, and Crystallographic Studies. |
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Journal, issue, pages | J. Am. Chem. Soc., Vol. 133, Page 16746-16749, Year 2011 |
Publish date | Jul 6, 2011 (structure data deposition date) |
![]() | Yao, Y. / Chen, P. / Diao, J. / Cheng, G. / Deng, L. / Anglin, J.L. / Prasad, B.V. / Song, Y. |
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Methods | X-ray diffraction |
Resolution | 2.5 Å |
Structure data | ![]() PDB-3sr4: |
Chemicals | ![]() ChemComp-TT8: ![]() ChemComp-GOL: ![]() ChemComp-ACT: ![]() ChemComp-SO4: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / HDOT1 / HISTONE LYSINE METHYLTRANSFERASE / TRANSFERASE-TRANSFERASE INHIBITOR complex |