+Search query
-Structure paper
Title | Unexpected binding orientation of bulky-B-ring anti-androgens and implications for future drug targets. |
---|---|
Journal, issue, pages | J. Med. Chem., Vol. 54, Page 3973-3976, Year 2011 |
Publish date | Apr 19, 2011 (structure data deposition date) |
Authors | Duke, C.B. / Jones, A. / Bohl, C.E. / Dalton, J.T. / Miller, D.D. |
External links | J. Med. Chem. / PubMed:21506597 |
Methods | X-ray diffraction |
Resolution | 1.7 - 1.9 Å |
Structure data | PDB-3rlj: PDB-3rll: |
Chemicals | ChemComp-RLJ: ChemComp-HOH: ChemComp-RLL: |
Source |
|
Keywords | TRANSCRIPTION / steroid receptor / DHT / testosterone |