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-Structure paper
Title | Structure-guided optimization of novel CDK2 inhibitors discovered by high-throughput screening |
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Journal, issue, pages | To be Published |
Publish date | Feb 2, 2011 (structure data deposition date) |
![]() | Schonbrunn, E. / Becker, A. / Betzi, S. / Alam, R. / Han, H. / Rawle, F. / Katta, V. / Jakkaraj, J. / Chakrasali, R. / Neelam, S. ...Schonbrunn, E. / Becker, A. / Betzi, S. / Alam, R. / Han, H. / Rawle, F. / Katta, V. / Jakkaraj, J. / Chakrasali, R. / Neelam, S. / Hook, D. / Tash, J. / Georg, G. |
![]() | Search PubMed |
Methods | X-ray diffraction |
Resolution | 1.6 - 2 Å |
Structure data | ![]() PDB-3ql8: ![]() PDB-3qqf: ![]() PDB-3qqg: ![]() PDB-3qqh: ![]() PDB-3qqj: ![]() PDB-3qql: ![]() PDB-3qrt: ![]() PDB-3qru: ![]() PDB-3qwj: ![]() PDB-3qwk: ![]() PDB-3qx2: ![]() PDB-3qx4: ![]() PDB-3qxo: ![]() PDB-3qzf: ![]() PDB-3qzg: ![]() PDB-3qzh: ![]() PDB-3qzi: ![]() PDB-3r1q: ![]() PDB-3r1s: ![]() PDB-3r1y: ![]() PDB-3r28: ![]() PDB-3r6x: ![]() PDB-3r71: ![]() PDB-3r73: ![]() PDB-3r7e: ![]() PDB-3r7i: ![]() PDB-3r7u: ![]() PDB-3r7v: ![]() PDB-3r7y: ![]() PDB-3r83: ![]() PDB-3r8l: ![]() PDB-3r8m: ![]() PDB-3r8p: ![]() PDB-3rai: ![]() PDB-3rm6: ![]() PDB-3rm7: ![]() PDB-3roy: ![]() PDB-3rpo: |
Chemicals | ![]() ChemComp-EDO: ![]() ChemComp-X01: ![]() ChemComp-HOH: ![]() ChemComp-X07: ![]() ChemComp-X06: ![]() ChemComp-PO4: ![]() ChemComp-X0A: ![]() ChemComp-X11: ![]() ChemComp-X03: ![]() ChemComp-X14: ![]() ChemComp-X19: ![]() ChemComp-X6A: ![]() ChemComp-X62: ![]() ChemComp-X63: ![]() ChemComp-X4B: ![]() ChemComp-X65: ![]() ChemComp-X66: ![]() ChemComp-X67: ![]() ChemComp-X69: ![]() ChemComp-X72: ![]() ChemComp-X75: ![]() ChemComp-X73: ![]() ChemComp-X76: ![]() ChemComp-XA0: ![]() ChemComp-X84: ![]() ChemComp-X86: ![]() ChemComp-X87: ![]() ChemComp-X88: ![]() ChemComp-X9I: ![]() ChemComp-X96: ![]() ChemComp-Z02: ![]() ChemComp-Z04: ![]() ChemComp-Z14: ![]() ChemComp-Z30: ![]() ChemComp-Z19: ![]() ChemComp-Z46: ![]() ChemComp-X85: ![]() ChemComp-18Z: ![]() ChemComp-19Z: ![]() ChemComp-22Z: ![]() ChemComp-24Z: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / protein kinase / inhibitor / TRANSFERASE-TRANSFERASE INHIBITOR complex |